AM251, Cannabinoid CB1 antagonist (TBI2007)
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AM251, Cannabinoid CB1 antagonist (TBI2007)
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Product Description
Description
Product Details
Formal Name: N-(Piperidin-1-yl)-5-(4-iodophenyl)-1-(2,4-dichlorophenyl)-4-methyl-1H-pyrazole-3-carboxamide
Molecular Formula: C22H21Cl2IN4O
Formula Weight: 555.24
CAS Number: 183232-66-8
Purity: >98%
Formulation: Powder
Solubility: Soluble in DMSO (up to 50 mg/ml) or in Ethanol (up to 13 mg/ml)
Storage: -20°C
Stability: ≥ 1 year.
Applications
Cannabinoid CB1 antagonist
Functions
A potent cannabinoid CB1 receptor antagonist with selectivity over CB2 receptors (306-fold). Displays anorectic effects and antidepressant-like effects in mice. Behaves as an agonist at GPR55, EC50=39nM. Active in vivo.
Application Procedures
First dissolved in DMSO (up to 50 mg/ml) or in Ethanol (up to 13 mg/ml), then diluted to aqueous buffer. Solutions in DMSO or ethanol may be stored at -20°C for up to 3 months.
